PKG drug G1

CAS No. 374703-78-3

PKG drug G1 ( —— )

Catalog No. M18488 CAS No. 374703-78-3

PKG drug G1 targets C42 of PKG Iα. PKG drug G1 can couple to vasodilation and blood pressure lowering by a C42 PKG Iα-independent mechanism.

Purity : 98%

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 46 In Stock
5MG 72 In Stock
10MG 110 In Stock
25MG 177 In Stock
50MG 335 In Stock
100MG 500 In Stock
500MG 1098 In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    PKG drug G1
  • Note
    Research use only, not for human use.
  • Brief Description
    PKG drug G1 targets C42 of PKG Iα. PKG drug G1 can couple to vasodilation and blood pressure lowering by a C42 PKG Iα-independent mechanism.
  • Description
    PKG drug G1 targets C42 of PKG Iα. PKG drug G1 can couple to vasodilation and blood pressure lowering by a C42 PKG Iα-independent mechanism.
  • Synonyms
    ——
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    PKG Iα
  • Research Area
    Cardiovascular Disease
  • Indication
    ——

Chemical Information

  • CAS Number
    374703-78-3
  • Formula Weight
    257.31
  • Molecular Formula
    C13H11N3OS
  • Purity
    98%
  • Solubility
    DMSO : ≥ 103 mg/mL; 400.30 mM
  • SMILES
    S=C3N/C(=C\c1c(C)nc2ccccc12)C(=O)N3
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Burgoyne JR, et al. Proof of Principle for a Novel Class of Antihypertensives That Target the Oxidative Activation of PKG Iα (Protein Kinase G Iα). Hypertension. 2017 Sep;70(3):577-586.
molnova catalog
related products
  • Kojibiose

    Kojibiose is a disaccharide in honey. Kojibiose is a product of the caramelization of glucose.

  • PAMBA

    4-(Aminomethyl)benzoic acid is an unnatural amino acid derivative, is an antifibrinolytic.

  • Dacisteine

    Dacisteine is an inhibitor of New Delhi metallo-beta-lactamase-1 (NDM-1, IC50 = 1000 μM).